DrLudovicaMonti

Barbosa da Silva E, Rocha DA, Fortes IS, Yang W, Monti L, Siqueira-Neto JL, Caffrey CR, McKerrow J, Andrade SF, Ferreira RSet al., 2021, Structure-Based Optimization of Quinazolines as Cruzain and <i>Tbr</i>CATL Inhibitors, Journal of Medicinal Chemistry, Vol: 64, Pages: 13054-13071, ISSN: 0022-2623

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Monti L, Cornec A-S, Oukoloff K, Kovalevich J, Prijs K, Alle T, Brunden KR, Smith AB, El-Sakkary N, Liu LJ, Syed A, Skinner DE, Ballatore C, Caffrey CRet al., 2021, Congeners Derived from Microtubule-Active Phenylpyrimidines Produce a Potent and Long-Lasting Paralysis of <i>Schistosoma mansoni</i> In Vitro, ACS Infectious Diseases, Vol: 7, Pages: 1089-1103, ISSN: 2373-8227

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Oukoloff K, Nzou G, Varricchio C, Lucero B, Alle T, Kovalevich J, Monti L, Cornec A-S, Yao Y, James MJ, Trojanowski JQ, Lee VM-Y, Smith AB, Brancale A, Brunden KR, Ballatore Cet al., 2021, Evaluation of the Structure–Activity Relationship of Microtubule-Targeting 1,2,4-Triazolo[1,5-<i>a</i>]pyrimidines Identifies New Candidates for Neurodegenerative Tauopathies, Journal of Medicinal Chemistry, Vol: 64, Pages: 1073-1102, ISSN: 0022-2623

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Ehrenkaufer G, Li P, Stebbins EE, Kangussu-Marcolino MM, Debnath A, White CV, Moser MS, DeRisi J, Gisselberg J, Yeh E, Wang SC, Company AH, Monti L, Caffrey CR, Huston CD, Wang B, Singh Uet al., 2020, Identification of anisomycin, prodigiosin and obatoclax as compounds with broad-spectrum anti-parasitic activity, PLOS Neglected Tropical Diseases, Vol: 14, Pages: e0008150-e0008150

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Monti L, Wang SC, Oukoloff K, Smith AB, Brunden KR, Caffrey CR, Ballatore Cet al., 2018, Brain-Penetrant Triazolopyrimidine and Phenylpyrimidine Microtubule Stabilizers as Potential Leads to Treat Human African Trypanosomiasis, ChemMedChem, Vol: 13, Pages: 1751-1754, ISSN: 1860-7179

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Lassalas P, Oukoloff K, Makani V, James M, Tran V, Yao Y, Huang L, Vijayendran K, Monti L, Trojanowski JQ, Lee VM-Y, Kozlowski MC, Smith AB, Brunden KR, Ballatore Cet al., 2017, Evaluation of Oxetan-3-ol, Thietan-3-ol, and Derivatives Thereof as Bioisosteres of the Carboxylic Acid Functional Group, ACS Medicinal Chemistry Letters, Vol: 8, Pages: 864-868, ISSN: 1948-5875

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Cornec A-S, Monti L, Kovalevich J, Makani V, James MJ, Vijayendran KG, Oukoloff K, Yao Y, Lee VM-Y, Trojanowski JQ, Smith AB, Brunden KR, Ballatore Cet al., 2017, Multitargeted Imidazoles: Potential Therapeutic Leads for Alzheimer’s and Other Neurodegenerative Diseases, Journal of Medicinal Chemistry, Vol: 60, Pages: 5120-5145, ISSN: 0022-2623

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Monti L, Stefanucci A, Pieretti S, Marzoli F, Fidanza L, Mollica A, Mirzaie S, Carradori S, De Petrocellis L, Schiano Moriello A, Benyhe S, Zádor F, Szűcs E, Ötvös F, Erdei AI, Samavati R, Dvorácskó S, Tömböly C, Novellino Eet al., 2016, Evaluation of the analgesic effect of 4-anilidopiperidine scaffold containing ureas and carbamates, Journal of Enzyme Inhibition and Medicinal Chemistry, Vol: 31, Pages: 1638-1647, ISSN: 1475-6366

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Morera E, Di Marzo V, Monti L, Allarà M, Schiano Moriello A, Nalli M, Ortar G, De Petrocellis Let al., 2016, Arylboronic acids as dual-action FAAH and TRPV1 ligands, Bioorganic &amp; Medicinal Chemistry Letters, Vol: 26, Pages: 1401-1405, ISSN: 0960-894X

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La Regina G, Coluccia A, Famiglini V, Pelliccia S, Monti L, Vullo D, Nuti E, Alterio V, De Simone G, Monti SM, Pan P, Parkkila S, Supuran CT, Rossello A, Silvestri Ret al., 2015, Discovery of 1,1′-Biphenyl-4-sulfonamides as a New Class of Potent and Selective Carbonic Anhydrase XIV Inhibitors, Journal of Medicinal Chemistry, Vol: 58, Pages: 8564-8572, ISSN: 0022-2623

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La Regina G, Bai R, Coluccia A, Famiglini V, Pelliccia S, Passacantilli S, Mazzoccoli C, Ruggieri V, Verrico A, Miele A, Monti L, Nalli M, Alfonsi R, Di Marcotullio L, Gulino A, Ricci B, Soriani A, Santoni A, Caraglia M, Porto S, Da Pozzo E, Martini C, Brancale A, Marinelli L, Novellino E, Vultaggio S, Varasi M, Mercurio C, Bigogno C, Dondio G, Hamel E, Lavia P, Silvestri Ret al., 2015, New Indole Tubulin Assembly Inhibitors Cause Stable Arrest of Mitotic Progression, Enhanced Stimulation of Natural Killer Cell Cytotoxic Activity, and Repression of Hedgehog-Dependent Cancer, Journal of Medicinal Chemistry, Vol: 58, Pages: 5789-5807, ISSN: 0022-2623

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