Publications
109 results found
Tyacke RJ, Robinson ESJ, Hume S, et al., 2004, Is P-glycoprotein responsible for the poor brain accumulation of the potential pet ligand BU97001 in rat brain?, Summer Meeting of the British-Association-for-Psychopharmacology, Publisher: SAGE PUBLICATIONS LTD, Pages: A35-A35, ISSN: 0269-8811
Robinson ESJ, Tyacke RJ, Finch L, et al., 2004, Pharmacological characterisation of novel α<sub>2</sub>-adrenoceptor antagonists as potential brain imaging agents, NEUROPHARMACOLOGY, Vol: 46, Pages: 847-855, ISSN: 0028-3908
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- Citations: 5
Glennon RA, Grella B, Tyacke RJ, et al., 2004, Binding of β-carbolines at imidazoline I<sub>2</sub> receptors:: a structure-affinity investigation, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, Vol: 14, Pages: 999-1002, ISSN: 0960-894X
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- Citations: 41
Chang-Fong J, Tyacke RJ, Lau A, et al., 2004, Pyrazino[1,2-<i>a</i>]indoles as novel high-affinity and selective imidazoline I<sub>2</sub> receptor ligands, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, Vol: 14, Pages: 1003-1005, ISSN: 0960-894X
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- Citations: 9
Glennon RA, Grella B, Tyacke RJ, et al., 2004, Binding of an imidazopyridoindole at imidazoline I<sub>2</sub> receptors, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, Vol: 14, Pages: 527-529, ISSN: 0960-894X
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- Citations: 12
Tyacke R, Robinson E, Hudson A, et al., 2004, Effects of endogenous noradrenaline on the <i>in vivo</i> binding of [<SUP>3</SUP>H]2-methoxyidazoxan ([<SUP>3</SUP>H]RX821002) in rat brain, 5th International Symposium on Functional Neuroreceptor Mapping of the Living Brain, Publisher: ACADEMIC PRESS INC ELSEVIER SCIENCE, Pages: T94-T95, ISSN: 1053-8119
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- Citations: 1
Tyacke RJ, Nutt DJ, Hudson AL, 2004, The relative affinities of (R)- and (S)-enantiomers of RX821002 the selective α2-adrenoceptor antagonist in rat whole brain, Winter Meeting
Abu Ghazaleh H, Lalies MD, Tyacke RJ, et al., 2004, Preliminary evaluation of the affinity of isoquinoline-containing compounds at imidazoline1 binding sites, Summer Meeting
Abu Ghazaleh H, Lalies MD, Tyacke RJ, et al., 2004, The structure-affinity relationship of BU98008 and its derivatives for imidazoline2 binding sites, Winter Meeting
Saczewski F, Hudson AL, Tyacke RJ, et al., 2003, 2-(4,5-Dihydro-1H-imidazol-2-yl)indazole (indazim) derivatives as selective I<sub>2</sub> imidazoline receptor ligands, EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, Vol: 20, Pages: 201-208, ISSN: 0928-0987
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- Citations: 31
Paterson L, Tyacke RJ, Robinson ESJ, et al., 2003, Role of monoamine oxidase in imidazoline<sub>2</sub> binding site mediated function in rat brain, 16th Congress of the European-College-of-Neuropsychopharmacology, Publisher: ELSEVIER SCIENCE BV, Pages: S104-S105, ISSN: 0924-977X
Tyacke RJ, Westaway J, Grella B, et al., 2003, Initial evaluation of two novel β-carbolines for rat brain imidazoline<sub>2</sub> binding sites, Summer Meeting of the British-Association-for-Psychopharmacology, Publisher: SAGE PUBLICATIONS LTD, Pages: A39-A39, ISSN: 0269-8811
Kimura A, Tyacke RJ, Minchin MCW, et al., 2003, Identification of a 55kDa imidazoline-2 binding protein in rabbit brain, Summer Meeting of the British-Association-for-Psychopharmacology, Publisher: SAGE PUBLICATIONS LTD, Pages: A38-A38, ISSN: 0269-8811
Kimura A, Tyacke RJ, Minchin MCW, et al., 2003, Identification of a putative imidazoline-2 binding protein, Meeting of the British-Pharmacological-Society-Clinical-Pharmacology-Section, Publisher: NATURE PUBLISHING GROUP, Pages: U87-U87, ISSN: 0007-1188
Tyacke RJ, Saçzewski F, Tabin P, et al., 2003, Initial evaluation of novel selective ligands for imidazoline<sub>2</sub> receptors in rat whole brain, AGMATINE AND IMIDAZOLINES: THEIR NOVEL RECEPTORS AND ENZYMES, Vol: 1009, Pages: 357-360, ISSN: 0077-8923
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- Citations: 1
Hudson AL, Tyacke RJ, Lalies MD, et al., 2003, Novel ligands for the investigation of imidazoline receptors and their binding proteins, AGMATINE AND IMIDAZOLINES: THEIR NOVEL RECEPTORS AND ENZYMES, Vol: 1009, Pages: 302-308, ISSN: 0077-8923
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- Citations: 21
Paterson LM, Tyacke RJ, Nutt DJ, et al., 2003, Relationship between imidazoline<sub>2</sub> sites and monoamine oxidase, AGMATINE AND IMIDAZOLINES: THEIR NOVEL RECEPTORS AND ENZYMES, Vol: 1009, Pages: 353-356, ISSN: 0077-8923
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- Citations: 7
Tyacke RJ, Lau A, Grella B, et al., 2003, Investigation of the affinities of two new β-carbolines for rat brain imidazoline<sub>2</sub> receptors, AGMATINE AND IMIDAZOLINES: THEIR NOVEL RECEPTORS AND ENZYMES, Vol: 1009, Pages: 361-363, ISSN: 0077-8923
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- Citations: 2
Kimura A, Tyacke RJ, Minchin MCW, et al., 2003, Identification of an I<sub>2</sub> binding protein from rabbit brain, AGMATINE AND IMIDAZOLINES: THEIR NOVEL RECEPTORS AND ENZYMES, Vol: 1009, Pages: 364-366, ISSN: 0077-8923
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- Citations: 6
Kimura A, Tyacke RJ, Nutt DJ, et al., 2002, Microautoradiography of imidazoline-2 binding sites in rabbit hypothalamus., Summer Meeting of the British-Association-for-Psychopharmacology, Publisher: SAGE PUBLICATIONS LTD, Pages: A63-A63, ISSN: 0269-8811
Paterson LM, Tyacke RJ, Nutt DJ, et al., 2002, The irreversible I<sub>2</sub> ligand BU99006 abolishes [<SUP>3</SUP>H]2BFI binding without effect on monoamine oxidase activity, Summer Meeting of the British-Association-for-Psychopharmacology, Publisher: SAGE PUBLICATIONS LTD, Pages: A63-A63, ISSN: 0269-8811
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- Citations: 2
Tyacke RJ, Davis N, Nutt DJ, et al., 2002, Initial evaluation of four potential imidazoline<sub>2</sub> pet ligands in rat whole brain, Summer Meeting of the British-Association-for-Psychopharmacology, Publisher: SAGE PUBLICATIONS LTD, Pages: A63-A63, ISSN: 0269-8811
Man J, Tyacke RJ, Saczewski F, et al., 2002, Initial evaluation of three novel selective ligands of imidazoline-2 receptors in rat whole brain, Summer Meeting of the British-Association-for-Psychopharmacology, Publisher: SAGE PUBLICATIONS LTD, Pages: A63-A63, ISSN: 0269-8811
Robinson ESJ, Tyacke RJ, Nutt DJ, et al., 2002, Distribution of [<SUP>3</SUP>H]BU224, a selective imidazoline I<sub>2</sub> binding site ligand, in rat brain, EUROPEAN JOURNAL OF PHARMACOLOGY, Vol: 450, Pages: 55-60, ISSN: 0014-2999
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- Citations: 15
Tyacke RJ, Robinson ESJ, Nutt DJ, et al., 2002, 5-Isothiocyanato-2-benzofuranyl-2-imidazoline (BU99006) an irreversible imidazoline<sub>2</sub> binding site ligand:: in vitro and in vivo characterisation in rat brain, NEUROPHARMACOLOGY, Vol: 43, Pages: 75-83, ISSN: 0028-3908
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- Citations: 15
Tyacke RJ, Robinson ESJ, Schnabel R, et al., 2002, N1′-fluoroethyl-naltrindole (BU97001) and N1′-fluorethyl-(14-formylamino)-naltrindole (BU97018) potential δ-opioid receptor PET ligands, NUCLEAR MEDICINE AND BIOLOGY, Vol: 29, Pages: 455-462, ISSN: 0969-8051
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- Citations: 9
Willmott G, Robinson ESJ, Tyacke RJ, et al., 2002, Functional characterisation of novel α<sub>2</sub>-adrenoceptor ligands in the mouse <i>vas deferens</i>, BRITISH JOURNAL OF PHARMACOLOGY, Vol: 135, ISSN: 0007-1188
Finch L, Tyacke RJ, Robinson ESJ, et al., 2002, <i>In vitro</i> evaluation of three potential SPECT ligands for the central α<sub>2</sub>-adrenoceptor, BRITISH JOURNAL OF PHARMACOLOGY, Vol: 135, ISSN: 0007-1188
Husbands SM, Glennon RA, Gorgerat S, et al., 2001, β-carboline binding to imidazoline receptors, DRUG AND ALCOHOL DEPENDENCE, Vol: 64, Pages: 203-208, ISSN: 0376-8716
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- Citations: 108
Robinson ESJ, Tyacke RJ, Nutt DJ, et al., 2001, Effect of BU99006, an irreversible imidazolme<sub>2</sub> binding site ligand, in the distribution of [<SUP>3</SUP>H]2BFI and of [<SUP>3</SUP>H]RX82I002 binding to rat brain sections, BRITISH JOURNAL OF PHARMACOLOGY, Vol: 133, Pages: U72-U72, ISSN: 0007-1188
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