BibTex format

author = {Azzarito, V and Rowell, P and Barnard, A and Edwards, TA and Macdonald, A and Warriner, SL and Wilson, AJ},
doi = {10.1002/cbic.201500504},
journal = {Chembiochem},
pages = {768--773},
title = {Probing Protein Surfaces: QSAR Analysis with Helix Mimetics},
url = {},
volume = {17},
year = {2016}

RIS format (EndNote, RefMan)

AB - α-Helix-mediated protein–protein interactions (PPIs) are important targets for small-molecule inhibition; however, generic approaches to inhibitor design are in their infancy and would benefit from QSAR analyses to rationalise the noncovalent basis of molecular recognition by designed ligands. Using a helix mimetic based on an oligoamide scaffold, we have exploited the power of a modular synthesis to access compounds that can readily be used to understand the noncovalent determinants of hDM2 recognition by this series of cell-active p53/hDM2 inhibitors.
AU - Azzarito,V
AU - Rowell,P
AU - Barnard,A
AU - Edwards,TA
AU - Macdonald,A
AU - Warriner,SL
AU - Wilson,AJ
DO - 10.1002/cbic.201500504
EP - 773
PY - 2016///
SN - 1439-7633
SP - 768
TI - Probing Protein Surfaces: QSAR Analysis with Helix Mimetics
T2 - Chembiochem
UR -
VL - 17
ER -